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RVX-208

Product Specifications

Background

RVX-208 is a potent BET bromodomain antagonist with IC50 of 0.510 μM for BD2, with approximately 170-fold selectivity over BD11,2. Increases apolipoprotein A-1 and HDL cholesterol in vitro and in vivo3. Reduces atherosclerosis4.

Conjugation

Unconjugated

Buffer

White solid

Storage Conditions

-20°C

Available Sizes

Frequently Asked Questions

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