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CID-2011756

Product Specifications

Background

Potent and selective ATP-competitive inhibitor of protein kinase D (PKD) . IC50=3.2, 0.6 and 0.7 μM for PKD1, 2 and 3 respectively. Inhibits phorbol ester-induced PKD activation in LNCaP prostate cancer cells. Cell permeable.

Conjugation

Unconjugated

Buffer

Tan solid

Storage Conditions

RT

Available Sizes

Frequently Asked Questions

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