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JNJ-1661010

Product Specifications

Background

Potent and selective FAAH inhibitor. Initially forms a covalent adduct with FAAH but is slowly released, IC50 = 12 nM. 100-fold selectivity for FAAH-1 over FAAH-2. Cell permeable and active in vivo. Displays analgesic activity in various animal models.

Conjugation

Unconjugated

Buffer

Off-white solid

Storage Conditions

-20°C

Available Sizes

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