Anagrelide HCl
Product Specifications
Background
Potent and selective phosphodiesterase (PDE3) inhibitor, IC50=36 nM) .1 Inhibits platelet production by disrupting megakaryocyte maturation2 via a mechanism which is independent of PDE3 inhibition3. Clinically useful agent for conditions requiring platelet lowering therapy.4,5
Conjugation
Unconjugated
Buffer
White solid
Storage Conditions
-20°C
Available Sizes
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