Pilsicainide (hydrochloride)

Pilsicainide hydrochloride (SUN-1165) is an orally active sodium channel blocker and potent class Ic antiarrhythmic agent[1][2].

Product Specifications

CAS Number

[88069-49-2]

Product Name Alternative

SUN-1165; Pilzicainide (hydrochloride)

UNSPSC

12352005

Hazard Statement

H301

Target

Sodium Channel

Type

Reference compound

Related Pathways

Membrane Transporter/Ion Channel

Applications

Neuroscience-Neuromodulation

Field of Research

Cardiovascular Disease

Assay Protocol

https://www.medchemexpress.com/pilsicainide-hydrochloride.html

Purity

99.94

Solubility

DMSO : 50 mg/mL (ultrasonic) |H2O : 100 mg/mL (ultrasonic)

Smiles

O=C(CC12N(CCC2)CCC1)NC3=C(C)C=CC=C3C.Cl

Molecular Formula

C17H25ClN2O

Molecular Weight

308.85

Precautions

H301

References & Citations

[1]Yamakawa M, et al. Effect of sodium channel blocker, pilsicainide hydrochloride, on net inward current of atrial myocytes in thyroid hormone toxicosis rats. Thyroid. 2005 Jul;15 (7) :653-9.|[2]Plosker GL. Pilsicainide. Drugs. 2010 Mar 5;70 (4) :455-67.