Setin-1
Setin-1 is one of the most potent inhibitors of Set7, acting by inhibiting KMTase G9a[1].
Product Specifications
CAS Number
[1313802-67-3]
UNSPSC
12352005
Target
Histone Methyltransferase
Type
Reference compound
Related Pathways
Epigenetics
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/setin-1.html
Smiles
FC(F)(C1=CC=C(C=C1)C2=CC=CC3=C2C=CN3C4=CC(CNC5=CC(C(O)=O)=CC=C5)=CC=C4)F
Molecular Formula
C29H21F3N2O2
Molecular Weight
486.48
References & Citations
[1]Kashyap S, et al. Using 'biased-privileged' scaffolds to identify lysine methyltransferase inhibitors. Bioorg Med Chem. 2014 Apr 1;22 (7) :2253-60.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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