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Enpp-1-IN-2

Enpp-1-IN-2 (Compound C) is a potent ENPP1 (ectonucleotide pyrophosphatase/phosphodiesterase 1) inhibitor with IC50 values of 0.26, 0.48 and 2.0 μM evaluated by means of TG-mAMP, pNP-TMP, and ATP assays, respectively. TG (Tokyo Green) -mAMP: a newly synthesized sensitive ENPP1 fluorescence probe[1].

Product Specifications

CAS Number

[2378640-92-5]

UNSPSC

12352005

Target

Phosphodiesterase (PDE)

Type

Reference compound

Related Pathways

Metabolic Enzyme/Protease

Applications

Cancer-programmed cell death

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/enpp-1-in-2.html

Purity

99.51

Solubility

DMSO : 100 mg/mL (ultrasonic)

Smiles

CC1=NC2=NC=NN2C(N(C)C)=C1CC3=CC=CC(N)=C3

Molecular Formula

C15H18N6

Molecular Weight

282.34

References & Citations

[1]Kawaguchi M, et al. Development of an ENPP1 Fluorescence Probe for Inhibitor Screening, Cellular Imaging, and Prognostic Assessment of Malignant Breast Cancer. J Med Chem. 2019 Oct 24;62 (20) :9254-9269.

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Available Sizes

Curated Selection

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