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TMX-4100

TMX-4100 is a selective phosphodiesterase 6D (PDE6D) degrader. TMX-4100 shows a high degradation preference for PDE6D with the DC50 values less than 200 nM in MOLT4, Jurkat, and MM.1S cells. TMX-4100 can be used for the research of multiple myeloma.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

262.29

Molecular Formula

C11H10N4O2S

Notes

Research use only, not for human use.

Receptor

Other Targets

CAS Number

2367619-63-2

Available Sizes

Curated Selection

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