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Picrotoxinin

Picrotoxinin is a blocker of chloride channel and a noncompetitive antagonist of GABAA with an IC50 of 1.15 μM for α1β2γ2L GABAA. Picrotoxinin shows convulsant properties.

Product Specifications

CAS Number

17617-45-7

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

292.3

Molecular Formula

C15H16O6

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

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