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Pep2m, myristoylated

Cell-permeable, myristoylated form of pep2m. Peptide inhibitor of the interaction between the C-terminus of the GluA2 (AMPA receptor) subunit and N-ethylmaleimide-sensitive fusion protein (NSF), a protein that regulates AMPA receptor function. Reduces postsynaptic currents in CA1 neurons, AMPA-mediated currents in cultured hippocampal neurons and AMPA receptor surface expression.

Product Specifications

CAS Number

1423381-07-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

1383.8

Molecular Formula

C63H118N18O14S

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

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