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RVD-Hpα

N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. Increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. Also high affinity CB2 positive allosteric modulator (Ki = 50 nM) .

Product Specifications

CAS Number

1193362-76-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

1424.66

Molecular Formula

C65H105N19O17

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

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