Tertiapin-Q
A high affinity blocker for inward-rectifier K+ channels, this compound is a stable derivative of the bee venom toxin tertiapin. Binds to ROMK1 (Kir1.1) and GIRK1/4 (Kir3.1/3.4) channels with high affinity (Ki values are 1.3 and 13.3 nM respectively) and is selective over Kir2.1 channels. Derivative tertiapin LQ also available.
Product Specifications
CAS Number
910044-56-3
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
2452
Molecular Formula
C106H175N35O24S4
Notes
Research use only, not for human use.
Receptor
——
Available Sizes
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