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ELA-21 (human)

High affinity apelin receptor agonist. Binds apelin receptors in left ventricle from normal and pulmonary arterial hypertensive (PAH) hearts (pKi values are 9.31 and 9.46, respectively) . Bioactive fragment of ELA-32. Inhibits forskolin-induced cAMP production and stimulates β-arrestin recruitment in vitro.

Product Specifications

CAS Number

2245073-05-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

2587.12

Molecular Formula

C112H184N40O25S3

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

Curated Selection

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