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AdTx1

Selective, high affinity, non-competitive α1A adrenoceptor antagonist (Ki = 0.35 nM) . Exhibits no significant activity against a range of other GPCRs, including α2A, β1 and β2 adrenoceptors. Antagonizes effects of phenylephrine on isolated rabbit prostate muscle in vitro and on intra-urethral pressure in rats.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

7283.22

Molecular Formula

C310H481N87O100S8

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

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