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Sar-[D-Phe8]-des-Arg9-Bradykinin

Potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant to aminopeptidase, kininase I and II (ACE) and neutral endopeptidase cleavage. Exhibits hypotensive and angiogenic activity in vivo.

Product Specifications

CAS Number

126959-88-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

975.11

Molecular Formula

C47H66N12O11

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

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