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FSLLRY-NH2

Selective PAR2 peptide antagonist. Reverses taxol-induced mechanical allodynia, heat hyperalgesia and PKC activation in ICR mice. Blocks ERK activation and collagen production in isolated cardiac fibroblasts. Also reduces symptoms in a mouse model of dermatophyte-associated itch.

Product Specifications

CAS Number

245329-02-6

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

796.97

Molecular Formula

C39H60N10O8

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

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