Des-His1-[Glu9]-Glucagon (1-29) amide
Glucagon receptor antagonist (pA2 = 7.2 for inhibition of glucagon-induced adenylyl cyclase activation in rat liver membranes) ; displays no agonist activity. Enhances glucose-stimulated pancreatic insulin release in vitro. Blocks added glucagon-induced hyperglycemia in normal rabbits without affecting glycogenolysis in vivo. Also blocks endogenous glucagon-induced hyperglycemia in streptozocin diabetic rats.
Product Specifications
CAS Number
110084-95-2
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
3358.68
Molecular Formula
C148H221N41O47S
Notes
Research use only, not for human use.
Receptor
——
Available Sizes
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