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JMV 449

Potent, metabolically stable neurotensin receptor agonist peptide (IC50 = 0.15 nM for inhibition of [125I]-NT binding to neonatal mouse brain; EC50 = 1.9 nM for contraction of guinea pig ileum) . Produces long-lasting hypothermic, neuroprotective and analgesic effects in mice following central administration in vivo.

Product Specifications

CAS Number

139026-66-7

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

746.96

Molecular Formula

C38H66N8O7

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

Curated Selection

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