MM 54
Potent apelin receptor antagonist (Ki = 82 nM; IC50 = 93 nM) . Antagonizes the inhibitory affect of [Pyr1]-Apelin-13 on forskolin-induced cAMP accumulation in CHO-K1-APJ cells. Recuces tumor expansion and lengthens survival time in a mouse xenograft model of glioblastoma.
Product Specifications
CAS Number
1313027-43-8
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
1737.15
Molecular Formula
C70H121N29O15S4
Notes
Research use only, not for human use.
Receptor
——
Available Sizes
Curated Selection
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