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[Phe1Ψ (CH2-NH) Gly2]Nociceptin (1-13) NH2

Potent agonist of the nociceptin (ORL1) receptor, demonstrated both in vitro and in vivo. Selective, competitive antagonism at the nociceptin receptor has also been reported (pA2 = 7.02 and 6.75 in the guinea pig ileum and mouse vas deferens respectively) .

Product Specifications

CAS Number

213130-17-7

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

1367.6

Molecular Formula

C61H102N22O14

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

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