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[ (pF) Phe4]Nociceptin (1-13) NH2

Highly potent and selective nociceptin/orphanin FQ receptor (OP4) agonist peptide (pKi = 10.68; pEC50 = 9.80) . Displays > 8000-fold selectivity over δ, κ, and μ opioid receptors and has relatively long lasting pronociceptive, hypotensive, negative inotropic and feeding stimulation effects in vivo.

Product Specifications

CAS Number

380620-88-2

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

1399.6

Molecular Formula

C61H99FN22O15

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

Curated Selection

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