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ProTx III

Potent Nav1.7 blocker (IC50 = 2.5 nM) . Also inhibits Nav1.1, Nav1.2, Nav1.3 and Nav1.6 in the nanomolar range. Exhibits no effects on Cav channels or nAChR at 5 μM. Demonstrates analgesic activity in vivo; antagonizes effects of scorpion-venom toxin OD1 at Nav1.7.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

3802.41

Molecular Formula

C162H246N52O43S6

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

Curated Selection

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