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BQ-3020 TFA (143113-45-5 free base)

BQ-3020 (TFA) is a selective ETB receptor agonist that inhibits [125I] et-1 binding to the ETB receptor in the cerebellum with a 0.2nm IC50, causing vasoconstriction.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

2120.35

Molecular Formula

C98H141F3N20O27S

Notes

Research use only, not for human use.

Receptor

IC50: 0.2 nM ([125I]ET-1 binding to ETB receptor)

Available Sizes

Curated Selection

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