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Urantide

Selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3) . Blocks hU-II induced contractions in thoracic aorta ex vivo. Exhibits no effect on noradrenaline or endothelin 1-induced contraction or on acetylcholine-induced relaxation. Behaves as a partial agonist in a calcium mobilization assay (in CHO cells expressing hUT receptors) .

Product Specifications

CAS Number

669089-53-6

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

1075.26

Molecular Formula

C51H66N10O12S2

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

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