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UFP 803

Urotensin-II (UT) receptor ligand; behaves as a silent antagonist in most in vitro assays and in vivo, but does retain small residual agonist activity under certain conditions in some assays. Competitively antagonizes U-II induced contractions in the rat aorta (pIC50 = 7.46) and prevents plasma extravasation elicited by U-II in mice in vivo.

Product Specifications

CAS Number

879497-82-2

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

1061.24

Molecular Formula

C50H64N10O12S2

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

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