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Exendin-3 (9-39) amide

Potent and selective GLP-1 receptor antagonist (Kd = 1.7 nM at cloned human GLP-1 receptors) . Inhibits cAMP production and insulin release induced by GLP-1 (7-36), exendin-3 (IC50 = 20 nM) and exendin-4. Blocks the inhibitory effect of GLP-1 on food intake in rats.

Product Specifications

CAS Number

133514-43-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

3369.79

Molecular Formula

C149H234N40O47S

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

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