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MCL 0020

Potent and selective melanocortin MC4 receptor antagonist (IC50 values are 11.63, 1115 and > 10 000 nM at MC4, MC3 and MC1 receptors respectively) . Significantly reverses stress-induced anorexia but has no effect on food intake in free-feeding rats. Exhibits anxiolytic-like activity in vivo.

Product Specifications

CAS Number

475498-26-1

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

609.73

Molecular Formula

C34H39N7O4

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

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