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Phrixotoxin 3

Potent blocker of voltage-gated sodium channels (IC50 values are 0.6, 42, and 72 nM for NaV1.2, NaV1.3 and NaV1.5 respectively) . Blocks inward sodium currents in a voltage-dependent manner.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

4059.74

Molecular Formula

C176H269N51O48S6

Notes

Research use only, not for human use.

Receptor

——

CAS Number

880886-00-0

Available Sizes

Curated Selection

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