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BI-2865

BI-2865 is a none-covalent pan-KRAS Inhibitor. BI-2865 binds to WT, G12C, G12D, G12V and G13D mutant KRAS with KDs of 6.9, 4.5, 32, 26, 4.3 nM respectively.

Product Specifications

CAS Number

2937327-93-8

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

465.57

Molecular Formula

C23H27N7O2S

Notes

Research use only, not for human use.

Receptor

——

Available Sizes

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