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SB-747651A Dihydrochloride

SB-747651A dihydrochloride is a chemical compound that serves as an ATP-competitive inhibitor for mitogen- and stress-activated kinase 1 (MSK1), featuring an IC50 of 11 nM. Additionally, this compound effectively inhibits PRK2, RSK1, p70S6K, and ROCK-II, showcasing its potential in inflammation research .

Product Specifications

CAS Number

1781882-72-1

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

415.32

Molecular Formula

C16H24Cl2N8O

Notes

Research use only, not for human use.

Receptor

ROCK

Available Sizes

Curated Selection

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