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LTGO-33

LTGO-33 is a species-specific inhibitor of the voltage-gated sodium channel NaV1.8, inhibiting NaV1.8, NaV1.1-NaV1.7, and NaV1.9.LTGO-33 inhibits wild-type and multiple NaV1.8 variants associated with human pain disorders and can be used for the study of pain.hBChE-IN-2 is a low affinity Nurr1 agonist.

Product Specifications

CAS Number

2834106-06-6

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

467.44

Molecular Formula

C21H17F4N3O3S

Notes

Research use only, not for human use.

Receptor

Sodium Channel

Available Sizes

Frequently Asked Questions

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