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UC-764864

UC-764864 is a selective UBE2N inhibitor that blocks E1-UBE2N thioester transfer, inhibits innate immune signaling and induces cytotoxic effects in MDS/AML cell lines and primary cells. In addition, UC-764864 reduces the ubiquitination status of UBE2N and can be used to study leukemia.

Product Specifications

CAS Number

278806-03-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

322.42

Molecular Formula

C19H18N2OS

Notes

Research use only, not for human use.

Receptor

E1/E2/E3 Enzyme

Available Sizes

Curated Selection

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