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Zamaporvint

Zamaporvint (RXC004) is a selective, orally active and potent inhibitor of the Wnt pathway that acts on the membrane-bound fatty acyltransferase porcupine to block Wnt ligand palmitoylation, secretion, and pathway activation.Zamaporvint has shown anti-tumor and anti-proliferative activity in a wide range of cancer cell lines.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

439.39

Molecular Formula

C21H16F3N7O

Notes

Research use only, not for human use.

Receptor

Others

CAS Number

1900754-56-4

Available Sizes

Curated Selection

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