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EN450

EN450 is a cysteine-responsive covalent molecular gel degrader of targeted NF-κB with antiproliferative and potentially anticancer activity, which acts through a dependence on Cullin E3 ligase and protease, and can be used to study leukemia.

Product Specifications

CAS Number

793719-01-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

288.75

Molecular Formula

C11H13ClN2O3S

Notes

Research use only, not for human use.

Receptor

NF-κB

Available Sizes

Curated Selection

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