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AXL-IN-13

AXL-IN-13 is a potent and orally active AXL inhibitor with an IC50 of 1.6 nM and a Kd of 0.26 nM. It exhibits anticancer activity, reverses TGF-β1-induced epithelial-mesenchymal transition (EMT), and inhibits cancer cell migration and invasion.

Product Specifications

CAS Number

2376928-82-2

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

632.72

Molecular Formula

C34H41FN6O5

Notes

Research use only, not for human use.

Receptor

FLT | PDGFR | TGF-beta/Smad | TAM Receptor

Available Sizes

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