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PARP10-IN-2

PARP10-IN-2 is a potent inhibitor of PARP10, a mono-ADP-ribosyltransferase, with an IC50 value of 3.64 μM for human PARP10. It also inhibits PARP2 and PARP15, with IC50 values of 27 μM and 11 μM, respectively.

Product Specifications

CAS Number

1042780-52-8

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

238.24

Molecular Formula

C14H10N2O2

Notes

Research use only, not for human use.

Receptor

PARP

Available Sizes

Curated Selection

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