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Palazestrant

Palazestrant (OP-1250) is an orally available and highly potent estrogen receptor antagonist and selective ER degrader with antitumor activity.Palazestrant inhibits 17b-estradiol (E2), inhibits MCF7 and CAMA-1 cell proliferation, and can be used in breast cancer research.

Product Specifications

CAS Number

2092925-89-6

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

449.6

Molecular Formula

C28H36FN3O

Notes

Research use only, not for human use.

Receptor

Estrogen/progestogen Receptor

Available Sizes

Frequently Asked Questions

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