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M3541

M3541 is a selectively potent and orally active ATM inhibitor with potential antitumor activity.M-3541 inhibits ATM kinase activity and ATM-mediated signaling by binding to ATM.M3541 prevents activation of DNA damage checkpoints, inhibits DNA damage repair, contributes to apoptosis, and induces death of ATM overexpressing tumor cells.

Product Specifications

CAS Number

1360628-91-6

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

428.42

Molecular Formula

C23H17FN6O2

Notes

Research use only, not for human use.

Receptor

Apoptosis | ATM/ATR

Available Sizes

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