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Bomedemstat ditosylate

Bomedemstat ditosylate (IMG-7289 ditosylate) is an orally active lysine-specific demethylase 1 (LSD1) inhibitor with antitumor activity that potentiates the response to PD-1 inhibition in a homozygous model of SCLC, inhibits cancer cell proliferation, and induces apoptosis. Bomedemstat ditosylate can be used to study myeloproliferative neoplasms and myelofibrosis.

Product Specifications

CAS Number

1990504-72-7

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

864.02

Molecular Formula

C42H50FN7O8S2

Notes

Research use only, not for human use.

Receptor

Apoptosis | Histone Demethylase

Available Sizes

Curated Selection

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