WDR5-0102
WDR5-0102 is a compound that inhibits the WDR5-MLL1 interface (K dis = 7 μM, K d = 4 μM), selectively reducing MLL1 HMT activity without affecting the human H3K4 methyltransferase SETD7 or other HMTs, including G9a, EHMT1, SUV39H2, SETD8, PRMT3, and PRMT5.
Product Specifications
CAS Number
824960-50-1
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
374.82
Molecular Formula
C18H19ClN4O3
Notes
Research use only, not for human use.
Receptor
Histone Methyltransferase
Available Sizes
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