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RBN-3143

RBN-3143 is a potent inhibitor of NAD+-competitive catalytic PARP14 (IC50= 4 nM), which inhibits ADP-ribosylation mediated by PARP14 and stabilizes PARP14 in cell lines, demonstrating research potential for lung inflammation.

Product Specifications

CAS Number

2360853-16-1

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

449.54

Molecular Formula

C22H28FN3O4S

Notes

Research use only, not for human use.

Receptor

PARP

Available Sizes

Curated Selection

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