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Vamotinib

Vamotinib (PF-114) is an orally active and specific tyrosine kinase inhibitor with antiproliferative and antitumour activity.Vamotinib inhibits the phosphorylation of BCR/ABL and BCR/ABL-T315I, which promotes apoptosis. Vamotinib is used to study drug-resistant Philadelphia chromosome-positive (Ph+) leukaemia and Alzheimer's disease.

Product Specifications

CAS Number

1416241-23-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

532.56

Molecular Formula

C29H27F3N6O

Notes

Research use only, not for human use.

Receptor

Bcr-Abl | Apoptosis | Tyrosine Kinases

Available Sizes

Frequently Asked Questions

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