Vamotinib
Vamotinib (PF-114) is an orally active and specific tyrosine kinase inhibitor with antiproliferative and antitumour activity.Vamotinib inhibits the phosphorylation of BCR/ABL and BCR/ABL-T315I, which promotes apoptosis. Vamotinib is used to study drug-resistant Philadelphia chromosome-positive (Ph+) leukaemia and Alzheimer's disease.
Product Specifications
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
532.56
Molecular Formula
C29H27F3N6O
Notes
Research use only, not for human use.
Receptor
Bcr-Abl | Apoptosis | Tyrosine Kinases
CAS Number
1416241-23-0
Available Sizes
Curated Selection
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