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GPR81 agonist 1

GPR81 agonist 1 is a potent and selective GPR81 agonist with high affinity for human and mouse GPR81, inhibiting lipolysis of differentiated 3T3-L1 adipocytes, improving insulin sensitivity and glycaemic control in mouse models of insulin resistance and diabetes, and can be used in the study of diabetes and obesity.

Product Specifications

CAS Number

1620992-67-7

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

446.63

Molecular Formula

C22H30N4O2S2

Notes

Research use only, not for human use.

Receptor

GPR

Available Sizes

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