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(R) -STU104

(R) -STU104 is a novel TAK1-MKK3 protein-protein interaction (PPI) inhibitor that inhibits TNF-α and suppresses the TAK1/MKK3/p38/MnK1/MK2/elF4E signalling pathway by binding to MKK3 and disrupting TAK1 phosphorylation of MKK3. (R) -STU104 is a candidate compound for the treatment of ulcerative colitis.

Product Specifications

CAS Number

2767124-77-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

298.33

Molecular Formula

C18H18O4

Notes

Research use only, not for human use.

Receptor

TNF | MAPK

Available Sizes

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