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IHMT-PI3Kδ-372 S-isomer

IHMT-PI3Kδ-372 S-isomer is a potent and selective PI3Kδ inhibitor with an IC50 of 14 nM. IHMT-PI3Kδ-372 S-isomer shows high selectivity over other class I PI3Ks (56∼83 fold) and other protein kinases. IHMT-PI3Kδ-372 can be uesd for chronic obstructive pulmonary disease (COPD) research.

Product Specifications

CAS Number

2429889-61-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

503.5

Molecular Formula

C26H23F2N7O2

Notes

Research use only, not for human use.

Receptor

PI3K

Available Sizes

Frequently Asked Questions

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