Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

PBRM1-BD2-IN-5

PBRM1-BD2-IN-5 is a potent inhibitor of the PBRM1 Bromodomain, with dissociation constant (Kd) values of 1.5 μM and 3.9 μM for PBRM1-BD2 and PBRM1-BD5 respectively, and an inhibitory concentration 50 (IC50) value of 0.26 μM for PBRM1-BD2. This compound effectively diminishes the interaction between full-length PBRM1 and acetylated histone peptide within the PBAF complex in cell lysates, making it a promising candidate for anticancer research.

Product Specifications

CAS Number

2819989-61-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

272.73

Molecular Formula

C15H13ClN2O

Notes

Research use only, not for human use.

Receptor

Epigenetic Reader Domain

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

HRP Linked Monoclonal Antibody to Complement Component 1, Q Receptor (C1qR1)
MBS2133080-01 0.1 mL

HRP Linked Monoclonal Antibody to Complement Component 1, Q Receptor (C1qR1)

Sign In for Pricing
View Details
HRP Linked Monoclonal Antibody to Complement Component 1, Q Receptor (C1qR1)
MBS2133080-02 0.2 mL

HRP Linked Monoclonal Antibody to Complement Component 1, Q Receptor (C1qR1)

Sign In for Pricing
View Details
HRP Linked Monoclonal Antibody to Complement Component 1, Q Receptor (C1qR1)
MBS2133080-03 0.5 mL

HRP Linked Monoclonal Antibody to Complement Component 1, Q Receptor (C1qR1)

Sign In for Pricing
View Details
HRP Linked Monoclonal Antibody to Complement Component 1, Q Receptor (C1qR1)
MBS2133080-04 1 mL

HRP Linked Monoclonal Antibody to Complement Component 1, Q Receptor (C1qR1)

Sign In for Pricing
View Details
HRP Linked Monoclonal Antibody to Complement Component 1, Q Receptor (C1qR1)
MBS2133080-05 5 mL

HRP Linked Monoclonal Antibody to Complement Component 1, Q Receptor (C1qR1)

Sign In for Pricing
View Details
HRP Linked Monoclonal Antibody to Complement Component 1, Q Receptor (C1qR1)
MBS2133080-06 5x 5 mL

HRP Linked Monoclonal Antibody to Complement Component 1, Q Receptor (C1qR1)

Sign In for Pricing
View Details