PBRM1-BD2-IN-2
PBRM1-BD2-IN-2, a selective and cell-active inhibitor of the polybromo-1 (PBRM1) bromodomain, exhibits binding affinity and inhibitory activity specifically targeting the PBRM1-BD2 domain, with Kd and IC50 values of 9.3 μM and 1.0 μM, respectively. This compound is utilized in cancer research.
Product Specifications
CAS Number
2819989-57-4
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
311.14
Molecular Formula
C14H9Cl2FN2O
Notes
Research use only, not for human use.
Receptor
Epigenetic Reader Domain
Available Sizes
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