What is the catalog number for GA-017?

The catalog number for GA-017 is M35303.

What sizes are available for GA-017?

GA-017 is available in the following size(s): 1 g, 500 mg, 5 mg, 10 mg, 25 mg, 50 mg, 100 mg, 200 mg.

How many pack sizes does GA-017 come in?

GA-017 is available in 8 different pack sizes.

GA-017 is currently made to order / not held in immediate stock. Contact us for lead time.

GA-017

GA-017 is a potent, selective inhibitor of LATS1 and LATS2 (large tumor suppressor kinase 1/2), exhibiting IC50 values of 4.10 and 3.92 nM, respectively. This compound simultaneously acts as an activator of cell proliferation by promoting YAP/TAZ activation and their nuclear translocation. Additionally, GA-017 enhances cell growth in 3D culture conditions and augments the ex vivo formation of mouse intestinal organoids .