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BMS202 hydrochloride (1675203-84-5 (free base) )

BMS202 hydrochloride (1675203-84-5 (free base) ) (PD-1/PD-L1 inhibitor 2 hydrochloride) is a small-molecule PD-1/PD-L1 interaction inhibitor (IC50: 18 nM) . Biophysical studies demonstrate that BMS202 binds directly to PD-L1. Binding of BMS202 promotes PD-L1 dimerisation and blocks the PD-L1/ PD1 interaction.

Product Specifications

CAS Number

2089334-95-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

455.97

Molecular Formula

C25H30ClN3O3

Notes

Research use only, not for human use.

Receptor

PD-1/PD-L1

Available Sizes

Curated Selection

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